Jul-Sep 1977;9(3):216-24. Ernest K. Mentioned compounds, studied on several species of animals, decrease blood pressure and the heart rate, modify catecholamine-induced effects, show properties characteristic for the beta-receptor blocking agents. Compounds of the general formula (1): Q1-Q2-C(=O)-N(R?1)-Q3-N(R2)-T1-Q4¿; and drugs which contain the compounds and are efficacious for thrombosis and embolism. This material is provided for educational purposes only and is not intended for medical advice, diagnosis or treatment. Phenolic ethylenediamine derivatives: a study of orally effective iron chelators. Drug Drug Description; Tripelennamine: A histamine H1 antagonist used to treat hypersensitivity reactions, coughs, and the common cold. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.) 2. Biochemical, morphochemical and pharmacodynamic evaluation of accumulation of ethylenediamine derivatives (ROM-203, MK-142) in some rat tissues. Benefit designs may vary with respect to drug coverage, quantity limits, days supply and prior authorization. Result indicated that the ethylenediamine derivatives, N,N-Bis(2-hydroxy-5-bromobenzyl)-1,2- ethanediamine (21), and N,N-Bis(2-hydroxy-5-chlorobenzyl)-1,2-ethanediamine (22) showed the most favorable antimicrobial activity exhibiting LC50 of 11.6 and 8.79 μM against S.enterica, 86 and 138 μM against P. aeruginosa, and 140 and 287 μM against S. aureus, respectively. Hershko C, Grady RW, Link G. Of 35 potential iron chelators screened for in vivo activity in rats, a group of phenolic compounds with excellent chelating properties were identified. Usually, PEG is converted to a carboxyl derivative and conju-gated with a protein as a simple acyl moiety. It is a bacteriostatic antimycobacterial drug, effective against Mycobacterium tuberculosis and some other mycobacteria. This formulary is subject to change throughout the year and plan exclusions may override this list. General pharmacological properties. We designed an amino acid type PEG (aaPEG) for preparation of a multi- ... A drug that binds to and activates gamma-aminobutyric acid receptors. ChemInform Abstract: ULTRA-SHORT-ACTING β-ADRENERGIC RECEPTOR BLOCKING AGENTS. Authors Leudimar … Allergy to ethylenediamine, Ethylenediamine allergy, Ethylenediamine dihydrochloride allergy, 1-2-Ethanediamine dihydrochloride allergy, 1-2-Diaminoethane dihydrochloride allergy, Chlorethamine allergy, C2H10Cl2N2 allergy. • These are clinically used in the treatment of histamine mediated allergic conditions like allergic rhinitis, allergic conjuctivitis etc., CLASSIFICATION: a) Amino alkyl ethers. View more via ChEBI Ontology . d) Phenothiazine derivatives… 1999 Mar;73(3):145-9. doi: 10.1016/s0162-0134(99)00009-4. Thioctic Acid ethylenediamine (a derivative of Thioctic Acid) is reported as an ingredient of Norstan Theophylline & Ethylenediamine in the following countries: South Africa; Important Notice: The Drugs.com international database is in BETA release. c) Propyl amine derivatives. DRUGS THAT BLOCK THE RELEASED HISTAMINE a) H1 ANTAGONISTS(FIRST GENERATION DRUGS): • These are classical antihistamines. Poly(amidoamine), or PAMAM, is a class of dendrimer which is made of repetitively branched subunits of amide and amine functionality.PAMAM dendrimers, sometimes referred to by the trade name Starburst, have been extensively studied since their synthesis in 1985, and represent the most well-characterized dendrimer family as well as the first to be commercialized. These drugs are often referred to simply as "piperazine" which may cause confusion between the specific anthelmintic drugs, the entire class of piperazine-containing compounds, and the compound itself. ethylenediamine derivatives heterocycle aromatic ring compounds general formula Prior art date 2000-04-05 Application number PCT/JP2001/002945 Other languages French (fr) Japanese (ja) Inventor Toshiharu Yoshino Tsutomu Nagata Noriyasu Haginoya Kenji Yoshikawa Hideyuki Kanno Masatoshi Nagamochi Original Assignee Daiichi Pharmaceutical Co., Ltd. Ethylenediamine-palladium(II) complexes with pyridine and its derivatives: synthesis, molecular structure and initial antitumor studies J Inorg Biochem . ethylenediamine: ChEBI ID CHEBI:30347: Definition An alkane-α,ω-diamine in which the alkane is ethane. [Pharmacological study of new ethylenediamine derivatives with antiarrhythmic activity]. Hydroxyethylethylenediamine is another commercially significant chelating agent. 2019 Oct 15;222:115002. doi: 10.1016/j.carbpol.2019.115002. This means it is still under development and may contain inaccuracies. Authoritative facts from DermNet New Zealand. b) Ethylenediamine derivatives. xH 2 O).As of 2015, the world hydrazine hydrate market amounted to $350 million. Triethylenetetramine (TETA and trien), also called trientine (), is an organic compound with the formula [CH 2 NHCH 2 CH 2 NH 2] 2.This oily liquid is colorless but, like many amines, assumes a yellowish color due to impurities resulting from air-oxidation.It is soluble in polar solvents. The pharmacology of new ethylenediamine derivatives (ROM-126, ROM-131, MK-142) with antiarrhythmic action. 3. Biochemical, morphochemical and pharmacodynamic evaluation of accumulation of ethylenediamine derivatives (ROM-203, MK-142) in some rat tissues Mater Med Pol. ethanolamine derivatives; ethylenediamine derivatives; first gen. antihist. All categories. derivatives, misc. Authors I Noyszewska-Skibińska, A … Ethylenediamine is an organic compound that is used as a building block for the production of many other chemical products. Drugs.com provides accurate and independent information on more than 24,000 prescription drugs, over-the-counter medicines and natural products. This drug entry is a stub and has not been fully annotated. [Article in Italian] Boni P, Bacciarelli C. PMID: 4442581 [PubMed - indexed for MEDLINE] Publication Types: English Abstract; MeSH Terms. Synthesis and Antimicrobial Evaluation of Amphiphilic Neamine Derivatives ... important antibiotics such as the natural drugs aminogly-cosides. Identification Name Ethylenediamine Accession Number DB14189 Description. ETHYLENEDIAMINE DERIVATIVES OF (ARYLOXY)PROPANOLAMINES HAVING ESTERS ON THE ARYL FUNCTION. substituted ethylenediamine ethylenediamine derivative derivative Prior art date 1983-12-01 Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.) It is also used as an excipient in many pharmacological preparations such as creams. Epub 2019 Jun 17. These compounds … Other uses The biochemical and antioxidant properties of chitosan modified with acetylacetone and ethylenediamine (Cacen) or diethylenetriamine (Cacdien) associated with ceftazidime (F) were investi … Biological properties of chitosan derivatives associated with the ceftazidime drug Carbohydr Polym. The design and synthesis of target compounds. PLEASE NOTE: Because prescription drug programs vary by group, the inclusion of a drug in this formulary does not imply coverage. It is scheduled to be annotated soon. Ethylenediamine derivatives possessing a substituent at the C1 position in S configuration and phenylenediamine derivatives possessing a substituent at the C5 position demonstrated moderate to strong anti-fXa activity. Title:2D Chemometrics Analyses of Tetrahydroquinoline and Ethylenediamine Derivatives with Antimalarial Activity VOLUME: 8 ISSUE: 2 Author(s): Humberto Fonseca de Freitas and Marcelo Santos Castilho Affiliation:Faculdade de Farmacia, Universidade Federal da Bahia (UFBA), Salvador, Bahia, 40170-115. Ethylenediamine (abbreviated as en when a ligand) is the organic compound with the formula C 2 H 4 (NH 2) 2.This colorless liquid with an ammonia-like odor is a strongly basic amine.It is a widely used building block in chemical synthesis, with approximately 500,000 tonnes produced in 1998. development of novel drug-carrier systems, although its sim-ple structure limits the types of hybrids that can be produced. Precursor to chelation agents, drugs, and agrochemicals A most prominent derivative of ethylenediamine is the chelating agent EDTA, which is derived from ethylenediamine via a Strecker synthesis involving cyanide and formaldehyde. antihistamine drugs. 2D Chemometrics Analyses of Tetrahydroquinoline and Ethylenediamine Derivatives with Antimalarial Activity. Data sources include IBM Watson Micromedex (updated 6 Jan 2021), Cerner Multum™ (updated 4 Jan 2021), ASHP … Chemischer Informationsdienst 1983, 14 (50) DOI: 10.1002/chin.198350126. ChEBI Name ethambutol: ChEBI ID CHEBI:4877: Definition An ethylenediamine derivative that is ethane-1,2-diamine in which one hydrogen attached to each of the nitrogens is sutstituted by a 1-hydroxybutan-2-yl group (S,S-configuration).It is a bacteriostatic antimycobacterial drug, effective against Mycobacterium tuberculosis and some other mycobacteria. Name Ethylenediamine Derivatives Accession Number DBCAT003721 Description Not Available Drugs. Drugs & Drug Targets. Part I. (14)C-Labeled ethylenediamine (EDA) was accumulated by slices of adult rat cerebral cortex, although the tissue:medium ratios were much lower than those for gamma-aminobutyric acid.EDA uptake was temp-dependent and appeared to take place by both sodium dependent and sodium independent mechanisms. ethylenediamine derivatives ethylenediamine derivatives Prior art date 2000-04-05 Application number ARP010101613A Other languages Spanish (es) Original Assignee Daiichi Seiyaku Co Priority date (The priority date is an assumption and is not a legal conclusion. Diethylcarbamazine, a derivative of piperazine, is used to treat some types of filariasis. Ethylenediamine Derivatives. February 2012; Medicinal chemistry (Shāriqah (United Arab Emirates)) 8(2):252-65 Inhibition studies indicate that ethylenediamine may be transported in part by the small … Ethambutol is an ethylenediamine derivative that is ethane-1,2-diamine in which one hydrogen attached to each of the nitrogens is sutstituted by a 1-hydroxybutan-2-yl group (S,S-configuration). Results and discussion 2.1. Studies J Inorg Biochem the date listed. drug, effective against tuberculosis... To and activates gamma-aminobutyric acid receptors performed a legal analysis and makes no representation as to the accuracy the. Description ; Tripelennamine: a study of orally effective iron chelators, ROM-131, MK-142 ) some! Medical advice, diagnosis or treatment Description not Available drugs vary with respect to drug,! Of accumulation of ethylenediamine derivatives: a study of new ethylenediamine derivatives ( ROM-203, MK-142 ) in some tissues... 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